- Induced fit versus conformational selection(2021)
Auteurs: Georges Vauquelin, Dominique Maes
- Fluxes for Unraveling Complex Binding Mechanisms(2020)
Auteurs: Georges Vauquelin, Dominique Maes, David C Swinney
Pagina's: 923-932
- Distinct in vivo target occupancy by bivalent- and induced-fit-like binding drugs(2017)
Auteurs: Georges Vauquelin
Pagina's: 4233-4246
- "Partial" competition of heterobivalent ligand binding may be mistaken for allosteric interactions: A comparison of different target interaction models(2015)
Auteurs: Georges Vauquelin, David Hall, Steven Charlton
Pagina's: 2300-2315
- Case study: Angiotensin receptor blockers (ARBs)(2015)
Series: Wiley's Methods and Principles in Medicinal Chemistry Series
Auteurs: Georges Vauquelin
Pagina's: 273-293
Aantal pagina's: 21
- Experimental Methods to Determine Binding Kinetics(2015)
Series: Wiley's Methods and Principles in Medicinal Chemistry Series
Auteurs: Georges Vauquelin, Walter Huber, David Swinney
Pagina's: 169-189
Aantal pagina's: 21
- Molecular mechanism of allosteric modulation: insight from a binding kinetics study at the human adenosine A1 receptor(2014)
Auteurs: D. Deval, , A. Massink, Van Velthoven Jpd, Georges Vauquelin, Ijzerman Ap, Heitman Lh
Pagina's: 5295-5312
- A study into the molecular mechanism of binding kinetics and long residence times of human CCR5 receptor antagonists(2014)
Auteurs: Swinney Davids, P. Beavis, Chuang Kt, Y. Zheng, I. Lee, P. Gee, J. Deval, Rotstein Dm, M. Dioszegi, P. Ravendran, et al.
Pagina's: 3364-3375
- Avidity and positive allosteric modulation/cooperativity act hand in hand to increase the residence time of bivalent receptor ligands.
doi: 10.1111/fcp.12052(2014)
Auteurs: Georges Vauquelin, Giampiero Bricca, Isabelle Van Liefde
Pagina's: 530-543
- [3H]IVDE77, a novel radioligand with high affinity and selectivity for the insulin-regulated aminopeptidase(2013)
Auteurs: Alexandros Nikolaou, Isabelle Van Den Eynde, Dirk Tourwé, Georges Vauquelin, Géza Tóth, Jayapal Reddy Mallareddy, Marko Poglitsch, Jo A Van Ginderachter, Patrick Vanderheyden
Pagina's: 93-102