Onderzoeker
Shrinivas Dumbre
- Disciplines:Ontdekking en evaluatie van biomarkers, Ontdekking en evaluatie van geneesmiddelen, Medicinale producten, Farmaceutica, Farmacognosie en fytochemie, Farmacologie, Farmacotherapie, Toxicologie en toxinologie, Andere farmaceutische wetenschappen, Bio-informatica en computationele biologie
Affiliaties
- Medicinale Chemie (Rega Instituut) (Afdeling)
Lid
Vanaf26 mrt 2007 → 30 sep 2019
Projecten
1 - 1 of 1
- Synthese, biologische evaluatie en conformationele studie van pentopyranoside nucleoside fosfonatenVanaf1 okt 2013 → 7 jun 2019Financiering: Eigen Middelen zoals patrimonium, inschrijvingsgelden, giften, ....
Publicaties
1 - 10 van 16
- Synthesis, conformational study and biological evaluation of pentopyranoside nucleoside phosphonates(2019)
Auteurs: Xiaochen Li, Piet Herdewyn, Shrinivas Dumbre
- Synthesis and Conformation of Pentopyranoside Nucleoside Phosphonates(2019)
Auteurs: Shrinivas Dumbre, Eveline Lescrinier, Elisabetta Groaz, Piet Herdewyn
Pagina's: 6589 - 6603 - Synthesis and structure-activity relationship studies of benzo[b][1,4]oxazin-3(4H)-one analogues as inhibitors of mycobacterial thymidylate synthase(2019)
Auteurs: Jakub Modranka, Nastia Parchina, Michiel Vanmeert, Shrinivas Dumbre, Roeland Vanhoutte, Jef Rozenski, Piet Herdewyn, Steven De Jonghe, Eveline Lescrinier
Pagina's: 645 - 662 - Kinetic analysis of N-alkylaryl carboxamide hexitol nucleotides as substrates for evolved polymerases.(2019)
Auteurs: Marleen Renders, Shrinivas Dumbre, Mikhail Abramov, Donaat Kestemont, Vitor Bernardes Pinheiro, Piet Herdewyn
Pagina's: 2160 - 2168 - Peptidoglycan glycosyltransferase-ligand binding assay based on tryptophan fluorescence quenching(2018)
Auteurs: Shrinivas Dumbre, Piet Herdewyn
Pagina's: 1 - 5 - Phosphonomethyl Oligonucleotides as Backbone-Modified Artificial Genetic Polymers(2018)
Auteurs: Jef Rozenski, Shrinivas Dumbre, Vitor Bernardes Pinheiro, Elisabetta Groaz, Piet Herdewyn
Pagina's: 6690 - 6699 - Threosyl nucleoside phosphonates as potential antiviral agents and constituents of artificial genetic systems(2017)
Auteurs: Chao Liu, Piet Herdewyn, Shrinivas Dumbre
- Synthesis and antiviral evaluation of base-modified deoxythreosyl nucleoside phosphonates(2017)
Auteurs: Chao Liu, Shrinivas Dumbre, Christophe Pannecouque, Steven De Jonghe, Piet Herdewyn
Pagina's: 5513 - 5528 - Synthesis of Polyhydroxylated Conidine Alkaloid as a Conformationally Restricted Azasugar(2016)
Auteurs: Shrinivas Dumbre
Pagina's: 2799 - 2802 - Amidate prodrugs of deoxythreosyl nucleoside phosphonates as dual inhibitors of HIV and HBV replication(2016)
Auteurs: Chao Liu, Shrinivas Dumbre, Christophe Pannecouque, Steven De Jonghe, Piet Herdewyn
Pagina's: 9513 - 9531