Targeting an aromatic hotspot in Plasmodium falciparum 1-deoxy-d-xylulose-5-phosphate reductoisomerase with U+03B2-arylpropyl analogues of fosmidomycin
Synthesis and evaluation of 1-deoxy-D-xylulose 5-phosphate reductoisomerase inhibitors as antimalarial and antituberculosis agents
Synthesis and evaluation of β-substituted fosmidomycin analogues as inhibitors of 1-deoxy-D-xylulose 5-phosphate reductoisomerase
Synthesis and bioactivity of U+03B2-substituted fosmidomycin analogues targeting 1-deoxy-D-xylulose-5-phosphate reductoisomerase
Synthetic fosmidomycin analogues with altered chelating moieties do not inhibit 1-deoxy-D-xylulose 5-phosphate reductoisomerase or Plasmodium falciparum growth in vitro