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Onderzoeker
Stijn Lenders
- Disciplines:Medicinale chemie
Affiliaties
- Medicinale Chemie (Rega Instituut) (Afdeling)
Lid
Vanaf10 sep 2019 → Heden
Projecten
1 - 1 of 1
- Ontwikkeling van nieuwe antimicrobiële middelen: Rationeel design van polyomavirus en mycobacteriële inhibitorenVanaf1 okt 2019 → 23 nov 2023Financiering: Eigen Middelen zoals patrimonium, inschrijvingsgelden, giften, ....
Publicaties
1 - 6 van 6
- Development of new antimicrobials: Rational design of polyomavirus and mycobacterial inhibitors(2023)
Auteurs: Stijn Lenders, Peter Verwilst, Sergei Strelkov, Arthur Van Aerschot
- Structural Basis of Cysteine Ligase MshC Inhibition by Cysteinyl-Sulfonamides(2022)
Auteurs: Stijn Lenders, Evgenii Osipov, Jef Rozenski, Sergei Strelkov, Arthur Van Aerschot
- Synthesis and structure-activity studies of novel anhydrohexitol-based Leucyl-tRNA synthetase inhibitors(2021)
Auteurs: Dries De Ruysscher, Luping Pang, Stijn Lenders, Jef Rozenski, Sergei Strelkov, Arthur Van Aerschot
- Facile Synthesis of Aminomethyl Phosphinate Esters as Serine Protease Inhibitors with Primed Site Interaction(2020)
Auteurs: Jan Pascal Kahler, Stijn Lenders, Merel van de Plassche, Steven Verhelst
Pagina's: 1739 - 1744 - Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction
Auteurs: Stijn Lenders
Pagina's: 3473 - 3517 - "Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction" (vol 65, pg 2204, 2022)
Auteurs: Stijn Lenders
Pagina's: 2204 - 2204