Extending the scope of the Aza-Fischer synthesis of 4- and 6-azaindoles

Fischer indole cyclization has recently been described as an efficient approach to the synthesis of azaindoles bearing electron-donating groups. We now show that this cascade reaction can be very efficient for the formation of a wider range of 4- and 6-azaindoles by using microwave irradiation.

Jaar van publicatie:2013

Trefwoorden:A1 Journal article

Toegankelijkheid:Closed