- Strecker-derived methodology for library synthesis of N-acylated alpha-aminonitriles(2021)
Auteurs: Pedro Goncalves, Anke Peeraer, Yves Adriaenssens, Lara Zonnekein, Philippe Franck, Bert Maes, Koen Augustyns, Pieter Van Der Veken
Pagina's: 1328 - 1338
- Caspase-3 probes for PET imaging of apoptotic tumor response to anticancer therapy(2019)
Auteurs: Tom Vanden Berghe, Yves Adriaenssens, Peter Vandenabeele, Koen Augustyns, Steven Staelens, Sigrid Stroobants, Pieter Van Der Veken, Leonie Wyffels
Pagina's: 4801 - 4824
- Carboxylate isosteres for caspase inhibitors(2017)
Auteurs: Yves Adriaenssens, D. Jiménez Fernández, L. Vande Walle, Filipe Elvas, Jurgen Joossens, Anne-Marie Lambeir, Koen Augustyns, M. Lamkanfi, Pieter Van Der Veken
Pagina's: 7456 - 7473
- Implementation of carboxylate isosteres to improve inflammatory caspase inhibitors(2017)
Auteurs: Yves Adriaenssens, Pieter Van Der Veken, Koen Augustyns
Aantal pagina's: 231
- Inhibitor screening and enzymatic activity determination for autophagy target Atg4B using a gel electrophoresis-based assay(2016)
Auteurs: Matthias Cleenewerck, Mandy Grootaert, Rafaela Gladysz, Yves Adriaenssens, Ria Roelandt, Jurgen Joossens, Anne-Marie Lambeir, Guido De Meyer, Wim Declercq, Koen Augustyns, et al.
Pagina's: 631 - 638
- Discovery and SAR of novel and selective inhibitors of urokinase plasminogen activator (uPA) with an imidazo[1,2-a]pyridine scaffold(2015)
Auteurs: Rafaela Gladysz, Yves Adriaenssens, Hans De Winter, Jurgen Joossens, Koen Augustyns, Pieter Van Der Veken
Pagina's: 9238 - 9257