Onderzoeker
Annelies Cannaert
- Trefwoorden:nieuw psychoactieve substanties, drug monitoring
- Disciplines:Analytische toxicologie, Klinische toxicologie, Forensische toxicologie
Affiliaties
- Vakgroep Bioanalyse (Departement)
Lid
Vanaf31 aug 2012 → 21 nov 2020
Projecten
1 - 3 of 3
- Het opsporen en profileren van opioïden in biologische matrices op basis van activiteit in plaats van structuur als alternatieve detectie methode in forensische toxicologie.Vanaf1 okt 2019 → 21 nov 2020Financiering: FWO junior postdoctoraal mandaat
- Screening op basis van activiteit in plaats van structuur van opioïden in biologische matrices als een nieuw concept in forensische toxicologie.Vanaf1 okt 2018 → 1 okt 2019Financiering: BOF - Nieuwe Onderzoeksinitiatieven
- Ontwikkeling van een snel een veelzijdig geneesmiddelen-reportersysteemVanaf1 jan 2013 → 31 dec 2016Financiering: IWT persoonsgebonden financ. - specialisatiebeurzen
Publicaties
1 - 10 van 35
- Off-target activity of NBOMes and NBOMe analogs at the mu opioid receptor(2023)
Auteurs: Marie Deventer, Mattias Persson, Antonio Laus, Eline Pottie, Annelies Cannaert, Graziella Tocco, Henrik Green
Pagina's: 1367 - 1384 - Are the N-demethylated metabolites of U-47700 more active than their parent compound? In vitro mu-opioid receptor activation of N-desmethyl-U-47700 and N,N-bisdesmethyl-U-47700(2022)
Auteurs: Frederike Nordmeier, Annelies Cannaert, Peter H. Schmidt, Markus R. Meyer, Nadine Schaefer
Pagina's: 713 - 717 - Machine learning to assist in large-scale, activity-based synthetic cannabinoid receptor agonist screening of serum samples(2022)
Auteurs: Liesl Janssens, Dimitri Boeckaerts, Simon Hudson, Daria Morozova, Annelies Cannaert, David M. Wood, Caitlin Wolfe, Bernard De Baets, Michiel Stock, Paul, I Dargan, et al.
Pagina's: 906 - 916 - Report on a new opioid NPS : chemical and in vitro functional characterization of a structural isomer of the MT-45 derivative diphenpipenol(2021)
Auteurs: Annelies Cannaert, Fabian Hulpia, Martijn Risseeuw, Katleen Van Uytfanghe, Eric Deconinck, Peter Blanckaert
Pagina's: 134 - 140 - Systematic evaluation of a panel of 30 synthetic cannabinoid receptor agonists structurally related to MMB-4en-PICA, MDMB-4en-PINACA, ADB-4en-PINACA, and MMB-4CN-BUTINACA using a combination of binding and different CB1 receptor activation assays-Part II: Structure activity relationship assessment via a beta-arrestin recruitment assay(2021)
Auteurs: Katharina Grafinger, Annelies Cannaert, Adam Ametovski, Eric Sparkes, Elizabeth Cairns, Samuel D. Banister, Volker Auwarter, Christophe Stove
Pagina's: 1402 - 1411 - The next generation of synthetic cannabinoids : detection, activity, and potential toxicity of pent-4en and but-3en analogues including MDMB-4en-PINACA(2021)
Auteurs: Alex J. Krotulski, Annelies Cannaert, Barry K. Logan
Pagina's: 427 - 438 - Systematic evaluation of a panel of 30 synthetic cannabinoid receptor agonists structurally related to MMB-4en-PICA, MDMB-4en-PINACA, ADB-4en-PINACA, and MMB-4CN-BUTINACA using a combination of binding and different CB1 receptor activation assays: Part I-Synthesis, analytical characterization, and binding affinity for human CB1 receptors(2021)
Auteurs: Edward Pike, Katharina Grafinger, Annelies Cannaert, Adam Ametovski, Jia Lin Luo, Eric Sparkes, Elizabeth A. Cairns, Ross Ellison, Roy Gerona, Volker Auwaerter, et al.
Pagina's: 1383 - 1401 - Systematic evaluation of a panel of 30 synthetic cannabinoid receptor agonists structurally related to MMB-4en-PICA, MDMB-4en-PINACA, ADB-4en-PINACA, and MMB-4CN-BUTINACA using a combination of binding and different CB1 receptor activation assays : part III : The G protein pathway and critical comparison of different assays(2021)
Auteurs: Katharina Elisabeth Grafinger, Marthe Vandeputte, Annelies Cannaert, Adam Ametovski, Eric Sparkes, Elizabeth Cairns, Patrick Osamu Juchli, Belal Haschimi, Benedikt Pulver, Samuel D. Banister, et al.
Pagina's: 1412 - 1429 - Diagnosing intake and rationalizing toxicities associated with 5F-MDMB-PINACA and 4F-MDMB-BINACA abuse(2021)
Auteurs: Wen Lie, Eleanor Jing Yi Cheong, Evelyn Mei Ling Goh, Hooi Yan Moy, Annelies Cannaert, Eric Chun Yong Chan
Pagina's: 489 - 508 - NNL-3 : a synthetic intermediate or a new class of hydroxybenzotriazole esters with cannabinoid receptor activity?(2021)
Auteurs: Adam Ametovski, Elizabeth A. Cairns, Katharina Elisabeth Grafinger, Annelies Cannaert, Marie Deventer, Shuli Chen, Xinyi Wu, Caitlin E. Shepperson, Felcia Lai, Ross Ellison, et al.
Pagina's: 4020 - 4036