Researcher
Pieter Annaert
- Disciplines:Biomarker discovery and evaluation, Drug discovery and development, Medicinal products, Pharmaceutics, Pharmacognosy and phytochemistry, Pharmacology, Pharmacotherapy, Toxicology and toxinology, Other pharmaceutical sciences
Affiliations
- Department of Pharmaceutical and Pharmacological Sciences (Department)
Responsible
From1 Aug 2020 → Today - Drug Delivery and Disposition (Division)
Member
From1 Oct 2005 → Today
Projects
1 - 10 of 33
- Investigating current gaps in time-dependent inhibition (TDI) and induction drug-drug interactions (DDIs). A focus on CYP3A4 and non-CYPs drug metabolizing enzymes (DMEs).From24 May 2023 → TodayFunding: Own budget, for example: patrimony, inscription fees, gifts
- Improved clearance prediction using ex vivo and new in silico tools to bridge the in vitro to in vivo extrapolation (IVIVE) gapFrom1 Oct 2022 → TodayFunding: Own budget, for example: patrimony, inscription fees, gifts
- Investigation of bidirectional pharmacokinetic drug-drug interaction between vicagrel, a novel analogue for the antiplatelet drug clopidogrel, and atorvastatinFrom15 Sep 2022 → TodayFunding: Own budget, for example: patrimony, inscription fees, gifts
- Design and development of FabV inhibitors as a new class of antibacterials for pathogenic Gram-negative bacteriaFrom1 Oct 2021 → TodayFunding: Baekeland
- Predicting exposure of neonates to maternal medicines via breastfeedingFrom1 Oct 2021 → TodayFunding: Own budget, for example: patrimony, inscription fees, gifts
- Model-informed drug development: application to drug-induced cholestasisFrom1 Oct 2021 → TodayFunding: Own budget, for example: patrimony, inscription fees, gifts
- Drug exposure through lactation: providing neonatal physiology to improve pharmacokinetic predictionsFrom21 Sep 2021 → TodayFunding: Own budget, for example: patrimony, inscription fees, gifts
- Drug Design and Development: From Target to MarketFrom7 Jun 2021 → TodayFunding: Own budget, for example: patrimony, inscription fees, gifts
- Integrated PK/PM Model-based Medication Dosing Assist App(lication) in KlinischWerkStation (KWS). Validation Studies of Tacrolimus in (Solid) Organ TransplantationFrom1 Jan 2021 → 31 Dec 2023Funding: IOF - technology validation in lab
- In vitro and in silico investigation of pharmacokinetics in neonates undergoing therapeutic hypothermiaFrom26 Nov 2020 → TodayFunding: Own budget, for example: patrimony, inscription fees, gifts
Publications
191 - 200 of 253
- Absorption characterization: the in situ intestinal perfusion technique in mice(2013)
Authors: Nico Holmstock, Patrick Augustijns, Pieter Annaert
- Exploring food effects on indinavir absorption with human intestinal fluids in the mouse intestine(2013)
Authors: Nico Holmstock, Tom De Bruyn, Jan Bevernage, Pieter Annaert, Jan Tack, Patrick Augustijns
Pages: 27 - 32 - Biorelevant in vitro evaluation of gastrointestinal drug supersaturation(2013)
Authors: Patrick Augustijns, Joachim Brouwers, Pieter Annaert
- Sandwich-cultured hepatocytes: utility for in vitro exploration of hepatobiliary drug disposition and drug-induced hepatotoxicity(2013)
Authors: Tom De Bruyn, Sagnik Chatterjee, Sarinj Fattah, Janneke Keemink, Johan Nicolaï, Patrick Augustijns, Pieter Annaert
Pages: 589 - 616 - HPLC-UV for detection of voriconazole in saliva samples(2013)
Authors: Kim Vanstraelen, Joachim Brouwers, Pieter Annaert, Patrick Augustijns, Ludo Willems, Isabel Spriet
Pages: 781 - 781 - Pharmacokinetic profile of voriconazole in a critically III patient on therapeutic plasma exchange(2013)
Authors: Isabel Spriet, Pieter Annaert, Philippe Meersseman, Eric Van Wijngaerden, Katrien Lagrou, Ludo Willems
Pages: 141 - 143 - Drug precipitation-permeation interplay: Supersaturation in an absorptive environment(2012)
Authors: Jan Bevernage, Joachim Brouwers, Pieter Annaert, Patrick Augustijns
Pages: 424 - 428 - Boosting of HIV protease inhibitors by ritonavir in the intestine: the relative role of Cyp and P-gp inhibition based on Caco-2 monolayers versus in situ intestinal perfusion in mice(2012)
Authors: Nico Holmstock, Pieter Annaert, Patrick Augustijns
Pages: 1473 - 1477 - Supersaturation in human gastric fluids(2012)
Authors: Jan Bevernage, Bart Hens, Joachim Brouwers, Jan Tack, Pieter Annaert, Patrick Augustijns
Pages: 184 - 189 - Nonclinical Testing Procedures-Pharmacokinetics(2012)
Authors: Pieter Annaert
Pages: 115 - 127