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Researcher
Nico Holmstock
- Disciplines:Biomarker discovery and evaluation, Drug discovery and development, Medicinal products, Pharmaceutics, Pharmacognosy and phytochemistry, Pharmacology, Pharmacotherapy, Toxicology and toxinology, Other pharmaceutical sciences
Affiliations
- Drug Delivery and Disposition (Division)
Member
From1 Oct 2008 → 7 Sep 2014
Projects
1 - 1 of 1
- Biopharmaceutical and pharmacokinetic factors determining the biological availibility of oral administrered HIV protease inhibitors.From1 Oct 2008 → 25 Feb 2013Funding: IWT personal funding - strategic basic research grants
Publications
1 - 7 of 7
- MRP2 inhibition by HIV protease inhibitors in rat and human hepatocytes: a quantitative confocal microscopy study(2018)
Authors: Nico Holmstock, Marlies Oorts, Pieter Annaert
Pages: 697 - 703 - Confocal imaging with a fluorescent bile acid analogue closely mimicking hepatic taurocholate disposition(2014)
Authors: Tom De Bruyn, Wouter Sempels, Nico Holmstock, Sagnik Chatterjee, Patrick Augustijns, Johan Hofkens, Hideaki Mizuno, Pieter Annaert
Pages: 1872 - 1881 - PXR/CYP3A4-humanized mice for studying drug-drug interactions involving intestinal P-glycoprotein(2013)
Authors: Nico Holmstock, Myriam Baes, Pieter Annaert, Patrick Augustijns
Pages: 1056 - 1062 - Absorption characterization: the in situ intestinal perfusion technique in mice(2013)
Authors: Nico Holmstock, Patrick Augustijns, Pieter Annaert
- Exploring food effects on indinavir absorption with human intestinal fluids in the mouse intestine(2013)
Authors: Nico Holmstock, Tom De Bruyn, Jan Bevernage, Pieter Annaert, Jan Tack, Patrick Augustijns
Pages: 27 - 32 - Boosting of HIV protease inhibitors by ritonavir in the intestine: the relative role of Cyp and P-gp inhibition based on Caco-2 monolayers versus in situ intestinal perfusion in mice(2012)
Authors: Nico Holmstock, Pieter Annaert, Patrick Augustijns
Pages: 1473 - 1477 - In situ intestinal perfusion in knockout mice demonstrates inhibition of intestinal P-glycoprotein by ritonavir causing increased darunavir absorption(2010)
Authors: Nico Holmstock, Pieter Annaert, Patrick Augustijns
Pages: 1407 - 1410