Researcher
Yves Depetter
- Disciplines:Transport phenomena, Other chemical sciences, Separation and membrane technologies, Process engineering, General chemical and biochemical engineering, Chemical product design and formulation, Catalysis and reacting systems engineering, Other (bio)chemical engineering, Agricultural plant production
Affiliations
- Department of Green Chemistry and Technology (Department)
Member
From1 Jan 2018 → 22 Sep 2019 - Department of Sustainable Organic Chemistry and Technology (Department)
Member
From19 Sep 2014 → 31 Dec 2017
Projects
1 - 1 of 1
- Design and development of new selective HDAC6 inhibitors with applications in cancer therapyFrom1 Oct 2014 → 14 Oct 2018Funding: BOF - Doctoral projects
Publications
1 - 9 of 9
- Expedient synthesis of lupulones and their derivatization to 2,8-7H-dihydrochromen-7-ones(2020)
Authors: Lena Decuyper, Gurkirat Kaur, Charlotte Versyck, Eline Blondeel, Yves Depetter, Kristof Van Hecke, Matthias D'hooghe
Pages: 442 - 444 - Selective pharmacological inhibitors of HDAC6 reveal biochemical activity but functional tolerance in cancer models(2019)
Authors: Yves Depetter, Rob De Vreese, Sophie Goethals, Elien Vandoorn, Alien Laevens, Jonas Steenbrugge, Pascal de Tullio, Marc Bracke, Matthias D'hooghe
Pages: 735 - 747 - Synthesis of indolineU+2010based benzhydroxamic acids as potential HDAC6 inhibitors(2019)
Authors: Yves Depetter, Jorick Franceus, Damijan Knez, Stanislav Gobec, Matthias D'hooghe
Pages: 12308 - 12312 - Synthesis of selective HDAC6 inhibitors and their evaluation in cancer models(2019)
Authors: Yves Depetter
- Assessment of the trifluoromethyl ketone functionality as an alternative zinc-binding group for selective HDAC6 inhibition(2018)
Authors: Yves Depetter, Flore Vanden Bussche, Rob De Vreese, Jorick Franceus, Matthias D'hooghe
Pages: 1011 - 1016 - Synthesis of potent and selective HDAC6 inhibitors bearing a cyclohexane- or cycloheptane-annulated 1,5-benzothiazepine scaffold(2017)
Authors: Rob De Vreese, Lisa Galle, Yves Depetter, Jorick Franceus, Kristof Van Hecke, Veronick Benoy, Ludo VanU+2005DenU+2005Bosch, Matthias D'hooghe
Pages: 128 - 136 - Synthesis and SAR assessment of novel Tubathian analogs in the pursuit of potent and selective HDAC6 inhibitors(2016)
Authors: Rob De Vreese, Yves Depetter, Tom Verhaeghe, Veronick Benoy, Wanda Haeck, Ludo Van Den Bosch, Matthias D'hooghe
Pages: 2537 - 2549 - Synthesis and anticancer properties of new (dihydro)pyranonaphthoquinones and their epoxy analogs(2015)
Authors: Anh Dang Thi Tuyet, Ha Vu Thi Thu, Thi Phuong Hoang, Ha Nguyen Thanh, Pham The Chinh, Vu Duc Cuong, Yves Depetter, Van Nguyen Tuyen, Matthias D'hooghe
Pages: 3355 - 3358 - Expedient stereoselective synthesis of new dihydropyrano- and dihydrofuranonaphthoquinones(2015)
Authors: Tuyet Anh Dang Thi, Yves Depetter, Karen Mollet, Hoang Thi Phuong, Doan Vu Ngoc, Chinh Pham The, Ha Thanh Nguyen, Thu Ha Nguyen Thi, Hung Huy Nguyen, Matthias D'hooghe, et al.
Pages: 2422 - 2425