Researcher
Belete Ayele Desimmie
- Disciplines:Microbiology, Systems biology, Laboratory medicine, Biomaterials engineering, Biological system engineering, Biomechanical engineering, Other (bio)medical engineering, Environmental engineering and biotechnology, Industrial biotechnology, Other biotechnology, bio-engineering and biosystem engineering
Affiliations
- Molecular Virology and Gene Therapy (Division)
Member
From3 Sep 2008 → 31 Mar 2013
Projects
1 - 1 of 1
- Novel HIV inhibitors targeting the interaction between integrase and LEDGF/p75From1 Sep 2008 → 12 Dec 2012Funding: BOF - Doctoral projects
Publications
1 - 10 of 16
- HIV-1 IN/Pol recruits LEDGF/p75 into viral particles(2015)
Authors: Belete Ayele Desimmie, Caroline Weydert, Rik Schrijvers, Sofie Vets, Jonas Demeulemeester, Paul Proost, Jan De Rijck, Rik Gijsbers, Frauke Christ, Zeger Debyser
- HIV-1 IN/Pol recruits LEDGF/p75 into viral particles(2015)
Authors: Belete Ayele Desimmie, Caroline Weydert, Rik Schrijvers, Sofie Vets, Jonas Demeulemeester, Paul Proost, Igor Paron, Jan De Rijck, Jan Mast, Norbert Bannert, et al.
Pages: 1 - 15 - Cellular cofactors as drug targets(2015)
Authors: Belete Ayele Desimmie, Frauke Christ, Zeger Debyser
Pages: 1 - 7 - Cellular cofactors as drug targets(2015)
Authors: Belete Ayele Desimmie, Frauke Christ, Zeger Debyser
Pages: 1 - 7 - Visceral Leishmaniasis Relapse in HIV Patients-A Role for Myeloid-Derived Suppressor Cells?(2014)
Authors: Belete Ayele Desimmie
- Validation of host factors of HIV integration as novel drug targets for anit-HIV therapy(2014)
Authors: Zeger Debyser, Belete Ayele Desimmie, Oliver Taltynov, Jonas Demeulemeester, Frauke Christ
Pages: 314 - 320 - 2-Hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs), novel inhibitors of HIV integrase with a high barrier to resistance(2013)
Authors: Belete Ayele Desimmie, Jonas Demeulemeester, Oliver Taltynov, Sergei Strelkov, Zeger Debyser, Frauke Christ
Pages: 1187 - 1194 - Rational design of LEDGINs as first allosteric integrase inhibitors for the treatment of HIV infection(2013)
Authors: Belete Ayele Desimmie, Jonas Demeulemeester, Frauke Christ, Zeger Debyser
Pages: e517 - e522 - LEDGINs inhibit late stage HIV-1 replication by modulating integrase multimerization in the virions(2013)
Authors: Belete Ayele Desimmie, Rik Schrijvers, Jonas Demeulemeester, Doortje Borrenberghs, Caroline Weydert, Sofie Vets, Johan Hofkens, Jan De Rijck, Jelle Hendrix, Rik Gijsbers, et al.
Pages: 57 - Phage display-directed discovery of LEDGF/p75 binding cyclic peptide inhibitors of HIV replication(2012)
Authors: Belete Ayele Desimmie, Eveline Lescrinier, Jelle Hendrix, Sofie Vets, Rik Gijsbers, Zeger Debyser, Frauke Christ
Pages: 2064 - 2075