Researcher
Bharat Gadakh
- Disciplines:Biomarker discovery and evaluation, Drug discovery and development, Medicinal products, Pharmaceutics, Pharmacognosy and phytochemistry, Pharmacology, Pharmacotherapy, Toxicology and toxinology, Other pharmaceutical sciences, Bioinformatics and computational biology
Affiliations
- Medicinal Chemistry (Rega Institute) (Division)
Member
From1 Sep 2010 → 31 Dec 2018
Projects
1 - 1 of 1
- Synthesis and biological evaluation of albomycin and aminoacyl sulfonamide analogues as potential aaRS inhibitors.From1 Oct 2015 → 30 Sep 2018Funding: FWO fellowships
Publications
1 - 10 of 16
- Design and synthesis of various nucleoside analogues as aminoacyl-tRNA synthetase inhibitors(2019)
Authors: Manesh Nautiyal, Arthur Van Aerschot, Stephen Weeks, Bharat Gadakh
- Family wide analysis of aminoacyl-sulfamoyl-3-deaza-adenosine analogues as inhibitors of aminoacyl-tRNA synthetases(2018)
Authors: Baole Zhang, Steff De Graef, Manesh Nautiyal, Luping Pang, Bharat Gadakh, Mathy Froeyen, Lieve Vanmellaert, Sergei Strelkov, Stephen Weeks, Arthur Van Aerschot
Pages: 384 - 396 - Different positions of amide side chains on the benzimidazo[1,2-: A] quinoline skeleton strongly influence biological activity(2018)
Authors: Sandra Liekens, Arthur Van Aerschot, Peter Vervaeke, Bharat Gadakh
Pages: 7096 - 7104 - Synthetic strategy and antiviral evaluation of diamide containing heterocycles targeting dengue and yellow fever virus(2016)
Authors: Joanna Zmurko, Suzanne Kaptein, Jef Rozenski, Bharat Gadakh, Patrick Chaltin, Arnaud Marchand, Johan Neyts, Arthur Van Aerschot
Pages: 158 - 168 - N-Acylated sulfonamide congeners of fosmidomycin lack any inhibitory activity against DXR(2015)
Authors: Bharat Gadakh, Jenny Pouyez, Johan Wouters, Akkaladevi Venkatesham, Paul Cos, Arthur Van Aerschot
Pages: 1577 - 9 - N-Acylated sulfonamide congeners of fosmidomycin lack any inhibitory activity against DXR(2015)
Authors: Bharat Gadakh, Arthur Van Aerschot
Pages: 1577 - 1579 - 5'-(N-aminoacyl)-sulfonamido-5'-deoxyadenosine: Attempts for a stable alternative for aminoacyl-sulfamoyl adenosines as aaRS inhibitors(2015)
Authors: Bharat Gadakh, Jef Rozenski, Mathy Froeyen, Arthur Van Aerschot
Pages: 227 - 236 - 5'-(N-aminoacyl)-sulfonamido-5'-deoxyadenosine: Attempts for a stable alternative for aminoacyl-sulfamoyl adenosines as aaRS inhibitors(2015)
Authors: Bharat Gadakh, Simon Smaers, Jef Rozenski, Mathy Froeyen, Arthur Van Aerschot
Pages: 227 - 36 - Renaissance in antibiotic discovery: some novel approaches for finding drugs to treat bad bugs(2015)
Authors: Bharat Gadakh, Arthur Van Aerschot
Pages: 2140 - 2158 - Renaissance in antibiotic discovery: some novel approaches for finding drugs to treat bad bugs(2015)
Authors: Bharat Gadakh, Arthur Van Aerschot
Pages: 2140 - 2158